Making Biliary Tract Cancer Treatment More Precise

Tumors arising in the gallbladder, bile ducts, and the small intestine are collectively referred to as biliary tract cancers. These cancers are rare—affecting approximately 12,350 individuals in 2024—but they are typically diagnosed at advanced stages when surgery, which can improve prognosis, is no longer an option.  Angela Lamarca, MD, PhD Systemic therapies, therefore, are the… Continue reading Making Biliary Tract Cancer Treatment More Precise

Discovery of isoquinoline-tethered quinazoline derivatives with enhanced HER2 inhibition over EGFR

Human epidermal growth factor receptor 2 (HER2) is a critical therapeutic target for HER2-positive or HER2-dependent cancers. While several HER2 kinase inhibitors have been identified, achieving high selectivity for HER2 over EGFR remains a significant challenge. In this study, we aimed to develop HER2-selective inhibitors with enhanced cellular activity. To improve the limited cellular activity… Continue reading Discovery of isoquinoline-tethered quinazoline derivatives with enhanced HER2 inhibition over EGFR

New dual-target therapy offers hope for better breast cancer treatment

Researchers, led by the University of Melbourne’s Professor Laura Mackay, a Laboratory Head and Immunology Theme Leader at the Peter Doherty Institute of Infection and Immunity (Doherty Institute), in collaboration with Pfizer, have discovered new insights into possible future treatments for breast cancer.  A new dual-target drug that has been shown to supercharge cancer-fighting immune… Continue reading New dual-target therapy offers hope for better breast cancer treatment

Estimating cancer incidence attributable to physical inactivity in the United States

Abstract Background Previous estimates of the number of cancers attributable to physical inactivity in the United States have typically focused on only three malignancies (colon, endometrial, and postmenopausal breast cancer). Contemporary epidemiologic evidence suggests that physical inactivity could contribute to up to 15 types of cancer, and a dose–response effect has been demonstrated for 13… Continue reading Estimating cancer incidence attributable to physical inactivity in the United States

Estimating cancer incidence attributable to physical inactivity in the United States

Abstract Background Previous estimates of the number of cancers attributable to physical inactivity in the United States have typically focused on only three malignancies (colon, endometrial, and postmenopausal breast cancer). Contemporary epidemiologic evidence suggests that physical inactivity could contribute to up to 15 types of cancer, and a dose–response effect has been demonstrated for 13… Continue reading Estimating cancer incidence attributable to physical inactivity in the United States

VP1-2025: Datopotamab deruxtecan (Dato-DXd) vs chemotherapy (CT) in previously-treated inoperable or metastatic hormone receptor-positive, HER2-negative (HR+/HER2–) breast cancer (BC): Final overall survival (OS) from the phase III TROPION-Breast01 trial

TROPION-Breast01 (NCT05104866) demonstrated statistically significant and clinically meaningful improvement in progression-free survival (PFS) by blinded independent central review (BICR) with the TROP2-directed ADC Dato-DXd vs investigator’s choice of CT (ICC) in patients (pts) with previously treated, inoperable/metastatic HR+/HER2– BC (HR 0.63 [95% CI 0.52–0.76]; p<0.0001). We report the final OS analysis and updated safety.